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BMS 986158
CAS No. 1800340-40-2
BMS 986158 ( BMS986158 )
Catalog No. M12735 CAS No. 1800340-40-2
BMS-986158 (BMS986158) is a potent and selective BET inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 245 | Get Quote |
|
| 10MG | 441 | Get Quote |
|
| 25MG | 707 | Get Quote |
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| 50MG | 972 | Get Quote |
|
| 100MG | 1314 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameBMS 986158
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NoteResearch use only, not for human use.
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Brief DescriptionBMS-986158 (BMS986158) is a potent and selective BET inhibitor.
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DescriptionBMS-986158 (BMS986158) is a potent and selective BET inhibitor, disrupts chromatin remodeling and prevents the expression of certain growth-promoting genes, resulting in an inhibition of tumor cell growth.Solid Tumors Phase 2 Clinical
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SynonymsBMS986158
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PathwayChromatin/Epigenetic
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TargetBromodomain
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RecptorBromodomain
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Research AreaCancer
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IndicationSolid Tumors
Chemical Information
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CAS Number1800340-40-2
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Formula Weight495.63
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Molecular FormulaC30H33N5O2
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Purity>98% (HPLC)
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SolubilityDMSO : 1 mg/mL 2.02 mM
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SMILESOC(C)(C)C1=CC=C2C(N([C@H](C3=CC=CC=C3)C4CCOCC4)C5=C2N=CC(C6=C(C)N=NN6C)=C5)=C1
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Chemical Name(S)-2-(3-(1,4-dimethyl-1H-1,2,3-triazol-5-yl)-5-(phenyl(tetrahydro-2H-pyran-4-yl)methyl)-5H-pyrido[3,2-b]indol-7-yl)propan-2-ol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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